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Metabolism and pharmacokinetics of the anti-HIV-1-specific inhibitor [1-[2′,5′-Bis-O-(tert-butyldimethylsilyl)-β-d-ribofuranosyl]-3-N-methyl-thymine]-3′-spiro-5″-(4″-amino-1″,2″-oxathiole-
Jan Balzarini; Lieve Naesens; Christina Bohman; Maria-Jésus Pérez-Pérez; Ana San-Félix; Maria-Jose Camarasa; Erik de Clercq
41
Synthesis of 3‘ ‘-Substituted TSAO Derivatives with Anti-HIV-1 and Anti-HIV-2 Activity through an Efficient Palladium-Catalyzed Cross-Coupling Approach
Lobatón; Esther; Rodríguez-Barrios; Fátima; Gago; Federico; Pérez-Pérez; María-Jesús; De Clercq; Erik; Balzarini; Jan; Camarasa; María-José; Velázquez; Sonsoles
43
Synthesis and Anti-HIV Activity of [AZT]-[TSAO-T] and [AZT]-[HEPT] Dimers as Potential Multifunctional Inhibitors of HIV-1 Reverse Transcriptase
Velazquez; Sonsoles; Alvarez; Rosa; San-Felix; Ana; Jimeno; Maria Luisa; De Clercq; Erik; Balzarini; Jan; Camarasa; Maria Jose