Terms search
1

Fluorination
Jinbo Hu; Teruo Umemoto
2

Studies on highly regio- and stereoselective fluorohydroxylation reaction of 3-aryl-1,2-allenyl phosphine oxides with Selectfluor
Guangke He; Chunling Fu; Shengming Ma
3

Copper mediated oxidation of amides to imides by Selectfluor
Zhuang Jin; Bo Xu; Gerald B. Hammond
4

Convenient fluorination of nitro and nitrile compounds with Selectfluor
Weimin Peng; Jean’ne M. Shreeve
5

An efficient green MCR protocol for the stereoselective synthesis of β-acetamido ketones catalyzed by Selectfluor™
V.S. Shinu; B. Sheeja; E. Purushothaman; D. Bahulayan
6

Oxidation of disulfides with Selectfluor™: concise syntheses of thiosulfonates and sulfonyl fluorides
Masayuki Kirihara; Sayuri Naito; Yuki Ishizuka; Honoka Hanai; Takuya Noguchi
7

A novel general method for preparation of α-fluoro-α-arylcarboxylic acid. Direct fluorination of silyl ketene acetals with Selectfluor®
Fei Zhang; Jake Z. Song
8

Straightforward access to tetrahydropyridine and piperidine-fused fluorolactones from pyridines and bis(trimethylsilyl)ketene acetals
Henri Rudler; Andrée Parlier; Louis Hamon; Patrick Herson; Patrick Chaquin; Jean-Claude Daran
9

Electrochemical monitoring of the oxidative coupling of alkynes catalyzed by triphenylphosphine gold complexes
Antonio Doménech; Antonio Leyva-Pérez; Saud I. Al-Resayes; Avelino Corma
10

Selectfluor-promoted fluorination of piperidinyl olefins
Meng-Yang Chang; Nien-Chia Lee; Ming-Fang Lee; Yu-Ping Huang; Chung-Han Lin
11

Halogenation of 1,1-diaryl alkenes
Meng-Yang Chang; Ming-Fang Lee; Chung-Han Lin; Nein-Chia Lee
12

Effect of acid catalysis on the direct electrophilic fluorination of ketones, ketals, and enamides using Selectfluor™
Jack Liu; Johann Chan; Craig M. Bryant; Petar A. Duspara; Ernest E. Lee; David Powell; Hua Yang; Ziping Liu; Chris Walpole; Edward Roberts; Robert A. Batey
13

Fluorine radical interception with radical traps: An experimental and DFT study
Xiang Zhang
14

Library-friendly synthesis of fluorinated ketones through functionalized hydration of alkynes and investigation of the reaction mechanism
Bo Xu; Weibo Wang; Gerald B. Hammond
15

Modern Gold Catalyzed Synthesis (TOSTE:GOLD_SYNTHESIS O-BK) || Gold-Catalyzed Oxygen-Atom Transfer to Alkynes
Hashmi; A. Stephen K.; Toste; F. Dean
16

Stereoselective Synthesis of Monofluoroalkyl α,β-Unsaturated Ketones From Allenyl Carbinol Esters Mediated by Gold and Selectfluor
Jin; Zhuang; Hidinger; Rachel S.; Xu; Bo; Hammond; Gerald B
17

Hydrogen abstraction/nucleophilic addition: A novel reaction pathway between aromatic olefin radical cation and TEMPO
Zhang Xiang
18

Sonochemical fluorination of heterocyclic nitro compounds with Selectfluor
Majid M. Sadeghi; Hossein Loghmani-Khouzani; Reza Ranjbar-Karimi; Philip Butler; Bernard T. Golding
19

Sonochemical fluorination of heterocyclic nitro compounds with Selectfluor™ (F-TEDA-BF4)
Majid M. Sadeghi; Hossein Loghmani-Khouzani; Reza Ranjbar-Karimi; Bernard T. Golding
20

Homogeneous gold-catalyzed efficient oxidative dimerization of propargylic acetates
Li Cui; Guozhu Zhang; Liming Zhang
21

One-pot fluorination followed by Michael addition or Robinson annulation for preparation of α-fluorinated carbonyl compounds
Yi; Wen-Bin; Huang; Xin; Cai; Chun; Zhang; Wei
22

Catalyst-free and highly selective electrophilic mono-fluorination of acetoacetamides: facile and efficient preparation of 2-fluoroacetoacetamides in PEG-400
Bi; Jingjing; Zhang; Zhiguo; Liu; Qingfeng; Zhang; Guisheng
23

Acceleration of alkenyltrimethylsilane fluorination under mild conditions using ultrasound
Reza Ranjbar-Karimi
24

Synthetic evolutions in the nucleophilic addition to alkynes
Bo Xu; Weibo Wang; Le-Ping Liu; Junbin Han; Zhuang Jin; Gerald B. Hammond
25

Synthesis of aryl allylic fluorides by direct electrophilic fluorination of alkenes
Hai-Qing Luo; Teck-Peng Loh
26

Thiophene and bioisostere derivatives as new MMP12 inhibitors
Matthew Badland; Delphine Compère; Karine Courté; Anne-Claude Dublanchet; Stéphane Blais; Ajith Manage; Guillaume Peron; Roger Wrigglesworth
27

Silver-Catalyzed Radical Phosphonofluorination of Unactivated Alkenes
Zhang; Chengwei; Li; Zhaodong; Zhu; Lin; Yu; Limei; Wang; Zhentao; Li; Chaozhong
28

One-pot synthesis of aryl fluorides by [3+3] cyclization of 1,3-bis(silyl enol ethers) with 2-fluoro-3-silyloxy-2-en-1-ones
Thomas Pundt; Matthias Lau; Ibrar Hussain; Mirza A. Yawer; Helmut Reinke; Peter Langer
29

Mono- and trifluorination of the thiazole ring of 2,5-diarylthiazoles using N-fluorobenzenesulfonimide (NFSI)
Hatfield; Julie M.; Eidell; Cheryl K.; Stephens; Chad E
30

Synthesis of 3-Amino-4-fluoropyrazoles
Surmont; Riccardo; Verniest; Guido; De Schrijver; Mathias; Thuring; Jan Willem; ten Holte; Peter; Deroose; Frederik; De Kimpe; Norbert
31

One-pot synthesis of α,α-difluoroimines from alkynes through tandem catalytic diboration/fluorination/imination reaction
Jesús Ramírez; Elena Fernández
32

Synthesis and heme-binding correlation with antimalarial activity of 3,6-bis-(ω-N,N-diethylaminoamyloxy)-4,5-difluoroxanthone
Rozalia A. Dodean; Jane X. Kelly; David Peyton; Gary L. Gard; Michael K. Riscoe; Rolf W. Winter
33

Two Metals Are Better Than One in the Gold Catalyzed Oxidative Heteroarylation of Alkenes
Tkatchouk; Ekaterina; Mankad; Neal P.; Benitez; Diego; Goddard; William A.; Toste; F. Dean
34

Chemo-enzymatic preparation of optically active thiiranes
Edyta Łukowska; Jan Plenkiewicz
35

Stereoselective fluorination of methylenecyclopropanes with N-F reagents: A modular entry to γ-fluorohomoallylic sulfonimides and γ-fluorohomoallylic amides
Weijun Fu; Guanglong Zou; Mei Zhu; Dongfeng Hong; Dongsheng Deng; Chen Xun; Baoming Ji
36

Bioactive fluorinated derivative of amphotericin B
Nobuaki Matsumori; Yuichi Umegawa; Tohru Oishi; Michio Murata
37

Synthesis and biological activity of brassinosteroids fluorinated at C-2
Sofía L. Acebedo; Javier A. Ramírez; Lydia R. Galagovsky
38

Regiospecific synthesis of α-chloro- and α-fluoro-1,2-diones
Riccardo Surmont; Bart De Corte; Norbert De Kimpe
39

α-Fluoro decalones as chiral epoxidation catalysts: fluorine effect
Arlette Solladié-Cavallo; Loïc Jierry; Arlette Klein; Michel Schmitt; Richard Welter
40

A new synthetic approach to 2,3-dideoxy-2-fluoro-β-d-threo-pentofuranose, the fluorofuranose unit of the anti-HIV-active nucleoside, β-FddA
Jean-Claude Caille; Hugues Miel; Paul Armstrong; M.Anthony McKervey
41

Copper(II) triflate-bis(oxazoline)-catalysed enantioselective electrophilic fluorination of β-ketoesters
Jun-An Ma; Dominique Cahard
42

Graphical contents list
43

A novel highly stereoselective multi-component synthesis of N-substituted β-amino ketone derivatives using copper(II) phthalocyanine as reusable catalyst
V.S. Shinu; P. Pramitha; D. Bahulayan
44

Discovery of TAK-733, a potent and selective MEK allosteric site inhibitor for the treatment of cancer
Qing Dong; Douglas R. Dougan; Xianchang Gong; Petro Halkowycz; Bohan Jin; Toufike Kanouni; Shawn M. O’Connell; Nicholas Scorah; Lihong Shi; Michael B. Wallace; Feng Zhou
45

InX3-catalyzed haloamidation of vinyl arenes: a facile synthesis of α-bromo- and α-fluoroamides
J.S. Yadav; B.V. Subba Reddy; D. Narasimha Chary; D. Chandrakanth
46

Synthesis and anti-HCV activity of a new 2′-deoxy-2′-fluoro-2′-C-methyl nucleoside analogue
Weidong Hu; Ping’an Wang; Chuanjun Song; Zhenliang Pan; Qiang Wang; Xiaohe Guo; Xuejun Yu; Zhenhua Shen; Shuyang Wang; Junbiao Chang
47

Synthesis and evaluation of 2′-substituted cyclobutyl nucleosides and nucleotides as potential anti-HIV agents
Yongfeng Li; Shuli Mao; Michael W. Hager; Kimberlynne D. Becnel; Raymond F. Schinazi; Dennis C. Liotta